A topical formamidine acaricide (tick and mite killer). It acts as an octopamine-receptor agonist in arthropod parasites (and has alpha-2 receptor agonist activity), causing over-stimulation and death of the parasite.

Drug class
Antiparasitics
Registered species
1
Recorded effects
0
Related products
1

Pharmacological information

A class-level scientific overview for general reference — no doses. The ultimate reference is always the locally approved product leaflet and consultation with a veterinarian.

Mechanism of action

A topical formamidine acaricide (tick and mite killer). It acts as an octopamine-receptor agonist in arthropod parasites (and has alpha-2 receptor agonist activity), causing over-stimulation and death of the parasite.

Indications

  • Mange (mites) and ticks in dogs, cattle, and pigs

Contraindications & warnings

  • Not to be used in horses — may cause colic and intestinal paralysis
  • Caution in cats, small dog breeds, and diabetic animals

Drug interactions

  • Its effects may be aggravated with monoamine oxidase inhibitors (MAOIs)
  • Its systemic (alpha-2) effect is reversed by alpha-2 antagonists such as atipamezole

Human-safety warning

Human hazard on ingestion or excessive skin exposure: may cause sedation and a fall in blood pressure. Wear gloves when handling and seek medical care upon accidental exposure.

Withdrawal periods

Note: Source: UK Veterinary Medicines Directorate (VMD). The figures are a guidance reference that may differ from the product registered in your country — always verify the locally approved leaflet and consult a veterinarian before slaughter or consuming products.
Apitraz 500 mg Bee-hive Strips for Honey Bees
Bee-hive strip · Laboratorios Calier, SA
SPC leaflet ↗
SpeciesMeatMilkEggs
Honey Bees———

Recorded adverse effects

openFDA veterinary reports — the numbers are report counts, not a severity rate.

No adverse-effect data recorded for this ingredient yet.

Sources